SCHEMBL8070833

SCHEMBL8070833

COc1ccnc(C[S+]([O-])c2nc3cc(N4CCN(C(=O)OC(C)(C)C)CC4)ccc3[nH]2)c1C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 6/20 0.40
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40
P2RX7 Q99572 1/20 0.39
SUV39H2 Q9H5I1 7/20 0.38
ABCB1 P08183 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
WNT3A P56704 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8075391 0.88 CCNT1 (0.42) ALKCCNT1CDK9GPR119PDE3B
SCHEMBL8074046 0.85 ATP1A1 (0.35) PDE3BPDE3AALDH1A1LMNAMAPT
SCHEMBL8069116 0.83 NPC1 (0.44) ALKCCNT1CDK9P2RX7SUV39H2
SCHEMBL8469710 0.79 ATP4A (0.37) ALDH1A1LMNAMAPT
Ilaprazole SCHEMBL23988478 0.78 ATP1A1 (0.36) ABCB1ALDH1A1LMNAMAPT
Ilaprazole SCHEMBL22734706 0.78 ATP1A1 (0.36) ABCB1ALDH1A1LMNAMAPT
Ilaprazole SCHEMBL22734704 0.78 ATP1A1 (0.36) ABCB1ALDH1A1LMNAMAPT
Ilaprazole SCHEMBL1179039 0.78 ATP1A1 (0.36) ABCB1ALDH1A1LMNAMAPT
SCHEMBL14467743 0.78 ATP4A (0.37)
Ilaprazole SCHEMBL8470106 0.77 ATP1A1 (0.36) ABCB1ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US claimed
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US disclosed
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed