SCHEMBL8071781

SCHEMBL8071781

Cc1ccc(-n2c(-c3ccc(S(N)(=O)=O)cc3)csc2=O)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.48
PTGS1 P23219 14/20 0.48
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA12 O43570 3/20 0.44
CA9 Q16790 3/20 0.44
CHRNA7 P36544 2/20 0.42
CA5A P35218 2/20 0.42
CA5B Q9Y2D0 2/20 0.42
PTGES O14684 1/20 0.41
HDAC3 O15379 1/20 0.41
PDPK1 O15530 1/20 0.41
PDE5A O76074 1/20 0.41
ABCB11 O95342 1/20 0.41
MT-CO2 P00403 1/20 0.41
LMNA P02545 1/20 0.41
CA3 P07451 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX5 P09917 1/20 0.41
ADORA3 P0DMS8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6723772 0.86 PTGS2 (0.39) PTGS2PTGS1CA1CA2CA12
SCHEMBL6733869 0.86 PTGS2 (0.35) PTGS2PTGS1CA1CA2CA12
SCHEMBL8071992 0.84 PTGS2 (0.51) PTGS2PTGS1CA1CA2CA12
SCHEMBL8061374 0.83 PTGS2 (0.61) PTGS2PTGS1CA1CA2CA12
SCHEMBL6725990 0.81 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL6722621 0.80 PTGS2 (0.38) PTGS2PTGS1CA1CA2CA12
SCHEMBL6732673 0.80 CA12 (0.33) PTGS2PTGS1CA1CA2CA12
SCHEMBL6732752 0.79 PTGS2 (0.36) PTGS2PTGS1CA1CA2CA12
SCHEMBL6726028 0.78 PTGS2 (0.36) PTGS2PTGS1CA1CA2CA12
SCHEMBL8061294 0.78 PTGS2 (0.52) PTGS2PTGS1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023277-A1 NOVEL 3,4-DIARYLTHIAZOLIN-2-ONE OR -2-THIONE DERIVATIVES, PREPARATION METHODS AND USES IN THERAPY LABORATOIRES UPSA (FR) 2000-08-02 EP claimed
WO-1999018093-A1 NOVEL 3,4-DIARYLTHIAZOLIN-2-ONE OR -2-THIONE DERIVATIVES, PREPARATION METHODS AND USES IN THERAPY LABORATOIRES UPSA (FR) 1999-04-15 WO claimed