SCHEMBL8072986

SCHEMBL8072986

CCOC(=O)c1ccc(CC(C)NCC(=O)c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.54
SIGMAR1 Q99720 1/20 0.53
DPP4 P27487 2/20 0.53
RAB9A P51151 4/20 0.50
NPC1 O15118 4/20 0.50
GAA P10253 1/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
ACACB O00763 1/20 0.48
ADRB1 P08588 2/20 0.47
ADRB3 P13945 1/20 0.47
USP2 O75604 2/20 0.47
CYP3A4 P08684 2/20 0.47
NR1I2 O75469 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
CHRM3 P20309 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10664191 0.81 ADRB3 (0.72) SMN1; SMN2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL9468493 0.80 ADRB3 (0.76) SMN1; SMN2ADRB1ADRB3ADRA1AALDH1A1
SCHEMBL9770881 0.79 SLC6A4 (0.54) SMN1; SMN2SIGMAR1RAB9ANPC1MEN1
SCHEMBL13417829 0.78 SMN1; SMN2 (0.54) SMN1; SMN2SIGMAR1RAB9ANPC1ACACB
SCHEMBL12326247 0.78 SMN1; SMN2 (0.54) SMN1; SMN2RAB9ANPC1GAAMEN1
SCHEMBL6541503 0.78 SMN1; SMN2 (0.58) SMN1; SMN2SIGMAR1GAAMEN1KMT2A
SCHEMBL9185848 0.77 SIGMAR1 (0.56) SMN1; SMN2SIGMAR1RAB9ANPC1CYP3A4
SCHEMBL19359211 0.77 SMN1; SMN2 (0.63) SMN1; SMN2RAB9ANPC1GAAMEN1
SCHEMBL8066591 0.76 SLC7A5 (0.59) SMN1; SMN2SIGMAR1DPP4RAB9ANPC1
Ethyl Benzoate SCHEMBL11244230 0.76 LMNA (0.68) SMN1; SMN2RAB9ANPC1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028080-A Quinolin-2-(1H)-ones MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-02-22 US disclosed
EP-0885196-A1 CHINOLINE-2-(1H)-ONES MERCK PATENT GmbH (DE) 1998-12-23 EP disclosed
WO-1997026244-A1 CHINOLINE-2-(1H)-ONES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-07-24 WO disclosed