Isoleucine

Isoleucine

SCHEMBL8073744

CCC(C)[C@@H](N)C(=O)O.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.50

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Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Isoleucine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.50
SLC1A2 P43004 1/20 0.50
SLC1A1 P43005 1/20 0.50
CA2 P00918 5/20 0.45
CA1 P00915 4/20 0.45
CYP2D6 P10635 1/20 0.44
MAPK1 P28482 1/20 0.44
DPP8 Q6V1X1 2/20 0.42
DPP9 Q86TI2 2/20 0.42
DPP7 Q9UHL4 1/20 0.42
GBA1 P04062 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoleucine SCHEMBL7996786 1.00 SLC1A3 (0.50) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL28869867 1.00 SLC1A3 (0.50) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL28279528 0.99 SLC1A3 (0.49) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL8048122 0.87 CA2 (0.44) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL8036374 0.87 CA2 (0.44) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL8036378 0.87 CA2 (0.44) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL8047310 0.87 CA2 (0.44) SLC1A3SLC1A2SLC1A1CA2CA1
Isoleucine SCHEMBL8047805 0.87 CA2 (0.44) SLC1A3SLC1A2SLC1A1CA2CA1
Valine SCHEMBL5159688 0.84 SLC1A3 (0.55) SLC1A3SLC1A2SLC1A1CA2CA1
Valine SCHEMBL2295611 0.84 SLC1A3 (0.55) SLC1A3SLC1A2SLC1A1CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028126-A1 DEPSIPEPTIDE DERIVATIVES BEARING PIPERAZINONE RINGS Nisshin Flour Milling Co., Ltd. (JP) 2000-08-16 EP disclosed