SCHEMBL8074148

SCHEMBL8074148

CCCc1ccc(C(O)c2ccc(F)cc2F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
F2RL1 P55085 3/20 0.41
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
PER2 O15055 1/20 0.37
CRY1 Q16526 1/20 0.37
CRY2 Q49AN0 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR7 P34969 1/20 0.36
LPL P06858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8075237 0.88 CYP3A4 (0.44) F2RL1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL1349957 0.82 CES2 (0.49) KMT2ACYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL8064702 0.77 KMT2A (0.40) KMT2ASLC6A2SLC6A4CES2CES1
SCHEMBL8064415 0.76 CYP3A4 (0.42) F2RL1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL4493580 0.76 DPP4 (0.44) KMT2ACYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL14814262 0.75 IDO1 (0.56) KMT2ACYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL30910880 0.75 IDO1 (0.56) KMT2ACYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL3909922 0.74 CES2 (0.55) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL21831133 0.71 F2RL1 (0.45) KMT2AF2RL1CYP3A4CYP2D6SLC6A2
SCHEMBL30910896 0.71 F2RL1 (0.45) KMT2AF2RL1CYP3A4CYP2D6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed