SCHEMBL8064702

SCHEMBL8064702

CCCc1ccc(C(O)c2cccc(F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
BRD4 O60885 2/20 0.40
CREBBP Q92793 1/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
LPL P06858 1/20 0.40
LIPG Q9Y5X9 1/20 0.40
OPRL1 P41146 3/20 0.39
OPRM1 P35372 2/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8064901 0.87 TSHR (0.42) BRD4CREBBPCES2CES1SLC6A2
SCHEMBL230519 0.79 CES2 (0.49) BRD4CES2CES1
SCHEMBL227352 0.79 CES2 (0.55) BRD4CES2CES1SLC6A2SLC6A4
SCHEMBL28788047 0.78 BRD4 (0.49) BRD4CREBBPCES2CES1OPRL1
SCHEMBL230487 0.77 IDO1 (0.52) BRD4CES2CES1SLC6A2SLC6A4
SCHEMBL8074148 0.77 KMT2A (0.42) KMT2ACES2CES1LPLLIPG
SCHEMBL8077592 0.76 CES2 (0.44) KMT2ABRD4CREBBPCES2CES1
SCHEMBL6349980 0.75 CES2 (0.45) BRD4CES2CES1OPRL1SLC6A2
SCHEMBL5169427 0.74 TAAR1 (0.57) LPLLIPGSLC6A4
SCHEMBL13849445 0.74 ESR1 (0.52) OPRM1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed