SCHEMBL8074149

SCHEMBL8074149

NC(=O)CCC(=O)c1cccc(Br)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.61
C1S P09871 1/20 0.52
ALDH1A1 P00352 2/20 0.49
GLA P06280 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HPGD P15428 2/20 0.46
GAA P10253 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ATM Q13315 1/20 0.44
NPC1 O15118 1/20 0.43
MGAM O43451 1/20 0.43
AMY1A P0DUB6 1/20 0.43
SI P14410 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035900 0.88 PARP1 (0.49) PARP1C1SALDH1A1GLASMN1; SMN2
SCHEMBL7403811 0.84 NR4A2 (0.62) PARP1ALDH1A1GLASMN1; SMN2GAA
SCHEMBL30666330 0.84 NR4A2 (0.62) PARP1ALDH1A1GLASMN1; SMN2GAA
SCHEMBL1814265 0.82 SMN1; SMN2 (0.56) PARP1ALDH1A1GLASMN1; SMN2HPGD
SCHEMBL3456365 0.81 L3MBTL1 (0.57) PARP1ALDH1A1GLASMN1; SMN2HPGD
SCHEMBL4518276 0.80 PARP1 (0.58) PARP1C1SALDH1A1GLASMN1; SMN2
SCHEMBL3357671 0.80 PARP1 (0.53) PARP1C1SALDH1A1GLASMN1; SMN2
SCHEMBL14277039 0.80 PARP1 (0.60) PARP1ALDH1A1SMN1; SMN2HPGDF2
SCHEMBL31149717 0.79 PARP1 (0.62) PARP1C1SALDH1A1GLASMN1; SMN2
SCHEMBL1808868 0.79 PARP1 (0.62) PARP1C1SALDH1A1GLASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6133302-A KYNURENINE-3-HYDROXYLASE ENZYME INHIBITORY ACTIVITY, AN ENZYME OF THE KYNURENINE (KYN) PATHWAY; COMPOUNDS SUCH AS 5-(3-(3-FLUOROPHENYL)-3-OXO-PROPYL)-1H-TETRAZOLE; FOR TREATMENT OF NEUROPATHOLOGICAL PROCESSES PHARMACIA & UPJOHN SPA (IT) 2000-10-17 US disclosed