SCHEMBL3357671

SCHEMBL3357671

O=C(CCCl)c1cccc(Br)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.53
ALDH1A1 P00352 3/20 0.50
GLA P06280 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.47
TP53 P04637 1/20 0.47
HPGD P15428 1/20 0.45
NPC1 O15118 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
MGAM O43451 1/20 0.44
AMY1A P0DUB6 1/20 0.44
GAA P10253 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
LMNA P02545 1/20 0.44
C1S P09871 1/20 0.44
RXFP1 Q9HBX9 1/20 0.43
RAB9A P51151 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1641363 0.89 PARP1 (0.50) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL3604586 0.88 PARP1 (0.49) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL13472220 0.86 L3MBTL1 (0.50) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL6390040 0.85 ALDH1A1 (0.57) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL3456365 0.83 L3MBTL1 (0.57) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL7403811 0.81 NR4A2 (0.62) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL30666330 0.81 NR4A2 (0.62) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL4518276 0.81 PARP1 (0.58) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL30758864 0.80 PARP1 (0.61) PARP1ALDH1A1GLAL3MBTL1TP53
SCHEMBL12139782 0.80 PARP1 (0.52) PARP1ALDH1A1GLAL3MBTL1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161272-A1 Phenanthrolines BASF SE (DE) 2010-03-10 EP disclosed
EP-2161272-A1 Phenanthrolines BASF SE (DE) 2010-03-10 EP disclosed
US-4025558-A SPIRO(CYCLOHEXANE-1,1*(2'H)-NAPHTHALENE); BENZOSPIRAN DERIVATIVES; CNS DEPRESSANTS, LOWERS BLOOD PRESSURE THE UPJOHN COMPANY (US) 1977-05-24 US disclosed
US-4010201-A AMINOBENZOSPIRANS, CENTRAL NERVOUS SYSTEM DEPRESSANT, HYPOTENSIVE THE UPJOHN COMPANY (US) 1977-03-01 US disclosed
US-3932425-A CNS DEPRESSANT, BLOOD PRESSURE LOWERING THE UPJOHN COMPANY (US) 1976-01-13 US disclosed