SCHEMBL8074204

SCHEMBL8074204

CCCC(c1cccc2c1C(=O)NC2=O)[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CASP3 P42574 6/20 0.34
GSK3B P49841 3/20 0.33
CASP2 P42575 1/20 0.33
CASP7 P55210 1/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
PARP1 P09874 1/20 0.33
CYP3A4 P08684 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
S100A4 P26447 2/20 0.31
PTPRC P08575 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1256987 0.77 KDM4E (0.40) POLBKDM4EALDH1A1GAAHPGD
SCHEMBL10731506 0.75 CYSLTR2 (0.39) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL9136212 0.75 ALDH1A1 (0.38) POLBKDM4EALDH1A1GAAHPGD
SCHEMBL6033869 0.75 KDM4E (0.38) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL10384426 0.74 KDM4E (0.40) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL11189703 0.73 ALDH1A1 (0.31) ALDH1A1GAACYP3A4TDP1MAPT
SCHEMBL28620531 0.73 KDM4E (0.37) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL30876940 0.73 KDM4E (0.43) POLBKDM4EALDH1A1GAAHPGD
SCHEMBL6285442 0.72 KDM4E (0.38) POLBKDM4EALDH1A1GAAHPGD
SCHEMBL4909210 0.72 ALDH1A1 (0.38) POLBKDM4EALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012165-A1 PROCESS FOR THE PREPARATION OF N-METHYL-D-PHENYLALANYL-N- 1- 3- (AMINOIMINOMETHYL)AMINO]PROPYL]-3,3-DIFLUORO-2-OXOHEXYL]-L-PROLINAMIDE Aventis Pharmaceuticals Inc. (US) 2000-06-28 EP disclosed
US-5739354-A ONE-STEP GUANYLATION OF 9,6-DIAMINO-5-HYDROXY-4,4-DIFLUORONONANE OR SALT; SIMPLIFICATION, HIGH YIELD END PRODUCT HOECHST MARION ROUSSEL, INC. (US) 1998-04-14 US disclosed
WO-1997035874-A1 PROCESS FOR THE PREPARATION OF N-METHYL-D-PHENYLALANYL-N-[1-[3-[(AMINOIMINOMETHYL)AMINO]PROPYL]-3,3-DIFLUORO-2-OXOHEXYL]-L-PROLINAMIDE HOECHST MARION ROUSSEL, INC. (US) 1997-10-02 WO disclosed