SCHEMBL8074642

SCHEMBL8074642

[2H]C([2H])([2H])C(C#N)(c1cc(C(=O)OC)cc(C(C#N)(C([2H])([2H])[2H])C([2H])([2H])[2H])c1)C([2H])([2H])[2H]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA12 O43570 3/20 0.43
CA7 P43166 3/20 0.43
CA9 Q16790 3/20 0.43
CA14 Q9ULX7 3/20 0.43
KDM4E B2RXH2 4/20 0.42
XDH P47989 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
NFKB1 P19838 1/20 0.42
GFER P55789 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
FUT7 Q11130 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL936288 0.90 NOTUM (0.46) NOTUMCA1CA2CA12CA7
SCHEMBL4199163 0.81 CA12 (0.58) NOTUMCA1CA2CA12CA7
SCHEMBL936865 0.81 CNR2 (0.43) NOTUMCA1CA2CA12CA7
SCHEMBL4200744 0.81 CA1 (0.43) NOTUMCA1CA2CA12CA7
SCHEMBL4969295 0.80 NOTUM (0.44) NOTUMCA1CA2CA12CA7
SCHEMBL5004408 0.80 ATAD2 (0.43) NOTUMCA1CA2CA12CA7
SCHEMBL4207015 0.80 NOTUM (0.63) NOTUMCA1CA2CA12CA7
SCHEMBL26146853 0.80 ALDH1A1 (0.42) NOTUMCA1CA2CA12CA7
SCHEMBL10187412 0.79 NOTUM (0.38) NOTUMCA1CA2CA12CA7
SCHEMBL5004975 0.77 NOTUM (0.41) NOTUMCA1CA2CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36617-E Anastrozole and salts as anticancer agent ZENECA LIMITED (GB) 2000-03-14 US disclosed
EP-0296749-B1 (Substituted aralkyl) heterocyclic compounds ZENECA LTD (GB) 1994-10-26 EP disclosed
US-4935437-A (Substituted aralkyl) heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-19 US disclosed
EP-0296749-A1 (Substituted aralkyl) heterocyclic compounds ZENECA LIMITED (GB) 1988-12-28 EP disclosed