SCHEMBL8075166

SCHEMBL8075166

C[C@H]1CCCc2ccc(C(N)=O)cc21

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 3/20 0.46
DRD2 P14416 2/20 0.46
KDM1A O60341 2/20 0.42
CYP3A4 P08684 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
OPRM1 P35372 4/20 0.40
ACHE P22303 2/20 0.40
OPRK1 P41145 2/20 0.39
KCNH2 Q12809 1/20 0.39
HSD17B3 P37058 1/20 0.38
OPRD1 P41143 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PARP10 Q53GL7 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25195403 0.88 AKR1C3 (0.44) DRD3DRD2KDM1AOPRM1OPRK1
SCHEMBL8080223 0.86 NPC1 (0.46) DRD3DRD2ACHEALDH1A1TAS1R3
SCHEMBL15235463 0.86 ALDH1A1 (0.54) DRD3KDM1AALDH1A1TAS1R3TAS1R1
SCHEMBL12620676 0.86 NPC1 (0.46) DRD3DRD2ACHEALDH1A1TAS1R3
SCHEMBL10175554 0.85 PARP10 (0.49) ACHEALDH1A1PARP10
Cyclohexane SCHEMBL8959188 0.84 NPC1 (0.45) DRD3DRD2ACHEALDH1A1TAS1R3
SCHEMBL15235464 0.82 KMT2A (0.45) ALDH1A1
SCHEMBL802970 0.82 ALDH1A1 (0.39) ACHEALDH1A1TAS1R3TAS1R1
SCHEMBL2227028 0.81 GNG2 (0.46) ACHE
SCHEMBL803415 0.78 ALDH1A1 (0.38) DRD3DRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009027601-A2 PYRAZOLE 3,5 CARBOXYLATE DERIVATIVES PREPARATION AND THERAPEUTIC APPLICATION THEREOF SANOFI-AVENTIS (FR) 2009-03-05 WO disclosed