SCHEMBL8075941

SCHEMBL8075941

C1=CC2CC1C(c1cccnc1)N2Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.51
MDM2 Q00987 1/20 0.51
ALDH1A1 P00352 3/20 0.42
KDM1A O60341 2/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
MAPT P10636 2/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
TRPV6 Q9H1D0 1/20 0.39
FPR1 P21462 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8072339 0.86 DRD4 (0.44) TP53MDM2ALDH1A1MAPTKDM4E
SCHEMBL8077458 0.83 CYP2A6 (0.40) ALDH1A1MAPK1KDM4E
SCHEMBL9058332 0.83 CYP2A6 (0.40) ALDH1A1MAPK1KDM4E
SCHEMBL8070733 0.75 CHRNB2 (0.46) ALDH1A1MAPT
SCHEMBL17598140 0.70 CHRM2 (0.45) ALDH1A1MAPTKDM4E
SCHEMBL9391377 0.70 CHRM2 (0.45) ALDH1A1MAPTKDM4E
SCHEMBL17598141 0.70 CHRM2 (0.45) ALDH1A1MAPTKDM4E
SCHEMBL24154837 0.69 KDM4E (0.42) ALDH1A1MAPTMAPK1KDM4E
SCHEMBL17585551 0.69 CHRM2 (0.44) ALDH1A1MAPTKDM4E
SCHEMBL17584402 0.68 CHRM2 (0.42) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100269-A ADMINISTERING TO PATIENT NICOTINIC RECEPTOR AGONISTIC DERIVATIVES OF 3-(PYRIDYL OR PYRIMIDYL)-2-AZABICYCLO(2.2.1) HEPTANE OR 2-AZABICYCLO(2.2.2.)OCTANE TO ELICIT NEUROTRANSMITTER SECRETION WITH REDUCED SIDE EFFECTS BENCHERIF MEROUANE (US) 2000-08-08 US disclosed
US-5583140-A ADMINISTERING 2-AZABICYCLO(2.2.2)OCT-5-ENE DERIVATIVES TO TREAT NEURODEGENERATIVE DISORDERS SUCH AS SENILE DEMENTIA OF ALZHEIMER'S TYPE TARGACEPT, INC. A CORP. OF DE, 1996-12-10 US disclosed
WO-1996036637-A1 PHARMACEUTICAL COMPOSITIONS FOR PREVENTION AND TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS R.J. REYNOLDS TOBACCO COMPANY (US) 1996-11-21 WO disclosed
WO-1996036637-A1 PHARMACEUTICAL COMPOSITIONS FOR PREVENTION AND TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS R.J. REYNOLDS TOBACCO COMPANY (US) 1996-11-21 WO disclosed