SCHEMBL8076201

SCHEMBL8076201

COc1cc2nc(N3CCN(c4nc(N)c(C(=O)O)nc4Cl)CC3)nc(N3CCNCC3)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 5/20 0.58
HPGD P15428 5/20 0.58
APAF1 O14727 1/20 0.58
POLB P06746 1/20 0.58
MAPT P10636 1/20 0.58
UBE2N P61088 1/20 0.58
WHR1 P49842 3/20 0.52
GLA P06280 3/20 0.46
HSD17B10 Q99714 3/20 0.46
MAPK1 P28482 2/20 0.46
GAA P10253 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
SLC22A1 O15245 1/20 0.46
ABCC4 O15439 1/20 0.46
LMNA P02545 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071848 0.85 TLR9 (0.60) KDM4EALDH1A1HPGDWHR1GLA
SCHEMBL8075717 0.84 WHR1 (0.42) KDM4EALDH1A1HPGDAPAF1POLB
SCHEMBL8076777 0.79 TLR9 (0.58) KDM4EALDH1A1HPGDWHR1GLA
SCHEMBL8784027 0.78 KDM4E (0.52) KDM4EALDH1A1HPGDAPAF1POLB
SCHEMBL8076773 0.78 KDM4E (0.42) KDM4EALDH1A1HPGDAPAF1POLB
Hydrochloric Acid SCHEMBL8786863 0.77 KDM4E (0.51) KDM4EALDH1A1HPGDAPAF1POLB
SCHEMBL20610675 0.77 ALDH1A1 (0.69) KDM4EALDH1A1HPGDAPAF1POLB
SCHEMBL8071627 0.76 TLR9 (0.53) KDM4EALDH1A1HPGDWHR1GLA
SCHEMBL20610678 0.76 ALDH1A1 (0.67) KDM4EALDH1A1HPGDAPAF1POLB
Aminodimethoxyquinazolinylpiperazine SCHEMBL32690190 0.75 KDM4E (1.00) KDM4EALDH1A1HPGDAPAF1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156758-A Antibacterial quinazoline compounds ISIS PHARMACEUTICALS, INC. (US) 2000-12-05 US disclosed