SCHEMBL8076996

SCHEMBL8076996

CC(=O)OC1C(Oc2ccnc(O)c2)c2cc(C#N)ccc2OC1(C)C

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 8/20 0.45
KDM4E B2RXH2 1/20 0.45
ABCB1 P08183 10/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324801 0.88 ABCC9 (0.43) ABCC9KDM4EABCB1CYP3A4
SCHEMBL7323149 0.86 ABCC9 (0.56) ABCC9KDM4EABCB1CYP3A4
SCHEMBL7331043 0.85 ABCC9 (0.46) ABCC9KDM4EABCB1
SCHEMBL7331226 0.82 ABCC9 (0.46) ABCC9KDM4EABCB1CYP3A4ALOX15
SCHEMBL8090760 0.77 KDM4E (0.40) ABCC9KDM4EABCB1CYP3A4ALOX15
SCHEMBL7325525 0.76 ABCB1 (0.39) ABCC9KDM4EABCB1
SCHEMBL8084932 0.76 ABCC9 (0.40) ABCC9KDM4EABCB1
SCHEMBL7328554 0.75 ABCC9 (0.39) ABCC9KDM4EABCB1
SCHEMBL7332368 0.75 ABCC9 (0.55) ABCC9KDM4EABCB1CYP3A4
SCHEMBL8088457 0.75 ABCC9 (0.40) ABCC9KDM4EABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed