SCHEMBL7328554

SCHEMBL7328554

CC1(C)CC(Oc2ccnc(O)c2)c2cc(C#N)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 10/20 0.39
ABCB1 P08183 3/20 0.39
SIRT2 Q8IXJ6 3/20 0.37
KDM4E B2RXH2 1/20 0.37
ABCC8 Q09428 2/20 0.36
KCNJ11 Q14654 2/20 0.36
KCNJ8 Q15842 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
SIRT1 Q96EB6 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326497 0.84 LMNA (0.33) KDM4ELMNA
SCHEMBL7321679 0.80 TLR3 (0.42) ABCC9SIRT2LMNA
SCHEMBL7325003 0.80 ABCC9 (0.40) ABCC9ABCB1SIRT2KDM4EABCC8
SCHEMBL7325525 0.80 ABCB1 (0.39) ABCC9ABCB1KDM4E
SCHEMBL7323149 0.80 ABCC9 (0.56) ABCC9ABCB1KDM4ECYP1A2CYP2D6
SCHEMBL7331043 0.79 ABCC9 (0.46) ABCC9ABCB1KDM4E
SCHEMBL8090760 0.77 KDM4E (0.40) ABCC9ABCB1KDM4ECYP1A2CYP2D6
SCHEMBL7333740 0.77 KDM4E (0.36) ABCC9ABCB1KDM4EABCC8KCNJ11
SCHEMBL8084932 0.76 ABCC9 (0.40) ABCC9ABCB1KDM4EABCC8KCNJ11
SCHEMBL8076996 0.75 ABCC9 (0.45) ABCC9ABCB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0363883-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1990-04-18 EP disclosed