SCHEMBL8078445

SCHEMBL8078445

CONNc1cccc(-c2nccs2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.47
PDPK1 O15530 1/20 0.47
CYP2A6 P11509 1/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP1B1 Q16678 1/20 0.43
SMPD3 Q9NY59 1/20 0.42
SYK P43405 2/20 0.41
ADRB2 P07550 1/20 0.40
KCNB1 Q14721 1/20 0.40
SRC P12931 1/20 0.40
CDK2 P24941 1/20 0.40
ZAP70 P43403 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
KAT6A Q92794 1/20 0.39
FFAR1 O14842 1/20 0.38
CFTR P13569 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355764 0.80 PDPK1 (0.55) EGFRPDPK1CYP2A6CYP1A1CYP1A2
SCHEMBL15606528 0.80 PDPK1 (0.58) EGFRPDPK1CYP2A6CYP1A1CYP1A2
SCHEMBL13994026 0.77 PDPK1 (0.50) EGFRPDPK1CYP2A6CYP1A1CYP1A2
SCHEMBL5216527 0.77 EGFR (0.52) EGFRPDPK1CYP2A6CYP1A1CYP1A2
SCHEMBL30849066 0.76 EGFR (0.55) EGFRPDPK1CYP2A6CYP1A1CYP1A2
SCHEMBL15805858 0.76 PDPK1 (0.72) EGFRPDPK1CYP2A6SMPD3ADRB2
SCHEMBL8083581 0.75 PRMT6 (0.48) CYP2A6
SCHEMBL8078588 0.75 PRMT6 (0.48) CYP2A6KAT6A
SCHEMBL29462071 0.74 DYRK1A (0.57) PDPK1CYP2A6CYP1A1CYP1A2CYP1B1
SCHEMBL1980934 0.74 DYRK1A (0.57) PDPK1CYP2A6CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836596-B1 HYDRAZINE DERIVATIVES UNIROYAL CHEM CO INC (US) 2000-08-23 EP disclosed
EP-0836596-A1 HYDRAZINE DERIVATIVES UNIROYAL CHEMICAL COMPANY, Inc. (US) 1998-04-22 EP disclosed
WO-1997002257-A1 HYDRAZINE DERIVATIVES UNIROYAL CHEMICAL COMPANY, INC. (US) 1997-01-23 WO disclosed