SCHEMBL8079404

SCHEMBL8079404

NC(N)=NCCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
CA12 O43570 2/20 0.57
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
CA9 Q16790 2/20 0.57
HTR3E A5X5Y0 1/20 0.56
HTR3B O95264 1/20 0.56
HTR3A P46098 1/20 0.56
HTR3D Q70Z44 1/20 0.56
HTR3C Q8WXA8 1/20 0.56
LOXL2 Q9Y4K0 1/20 0.52
PLAU P00749 1/20 0.51
IDO1 P14902 4/20 0.50
KCNJ1 P48048 2/20 0.47
F2 P00734 1/20 0.47
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
KCNH2 Q12809 1/20 0.47
ALDH1A1 P00352 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004498 0.77 TSHR (0.55) TSHRCA12CA1CA2CA9
SCHEMBL2850348 0.77 TSHR (0.59) TSHRLOXL2IDO1KCNJ1KCNH2
SCHEMBL18913824 0.77 TSHR (0.69) TSHRLOXL2IDO1KCNJ1KCNH2
SCHEMBL30758863 0.77 TSHR (0.69) TSHRLOXL2IDO1KCNJ1KCNH2
Sulfuric Acid SCHEMBL10890618 0.77 F2 (0.53) TSHRCA12CA1CA2CA9
SCHEMBL3292782 0.77 TSHR (0.75) TSHRLOXL2IDO1KCNJ1KCNH2
SCHEMBL6821944 0.76 TSHR (0.58) TSHRLOXL2IDO1KCNJ1KCNH2
SCHEMBL530075 0.75 TSHR (0.61) TSHRLOXL2IDO1KCNJ1KCNH2
SCHEMBL43299 0.74 LOXL2 (0.64) TSHRLOXL2IDO1KCNJ1KCNH2
SCHEMBL1119530 0.74 TSHR (0.60) TSHRLOXL2IDO1KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882066-B1 PEPTIDE DERIVATIVES ZENECA LTD (GB) 2000-09-06 EP disclosed
US-6087336-A ANTIINFLAMMATORY AGENT TREATING RHEUMATOID ARTHRITIS ZENECA LIMITED (GB) 2000-07-11 US disclosed
EP-0882066-A1 PEPTIDE DERIVATIVES ZENECA LIMITED (GB) 1998-12-09 EP disclosed
WO-1997031023-A1 PEPTIDE DERIVATIVES ZENECA LIMITED (GB) 1997-08-28 WO disclosed