SCHEMBL807987

SCHEMBL807987

CC(C)(N)c1ccc(-c2nnc3cnc4ccc(-c5ccc6[nH]ncc6c5)cc4n23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.38
ROCK2 O75116 4/20 0.38
AURKB Q96GD4 3/20 0.38
PIM1 P11309 2/20 0.38
QPCT Q16769 1/20 0.38
QPCTL Q9NXS2 1/20 0.38
CLK1 P49759 2/20 0.38
DYRK3 O43781 1/20 0.38
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
CDK5 Q00535 1/20 0.38
DYRK1A Q13627 1/20 0.38
CDK5R1 Q15078 1/20 0.38
DYRK2 Q92630 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
TRPA1 O75762 2/20 0.38
MAPKAPK2 P49137 1/20 0.37
PRKCH P24723 1/20 0.37
PRKCQ Q04759 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807837 0.89 PRKDC (0.38) PIK3CAPIK3CBPRKDCATRATRIP
SCHEMBL15133602 0.88 MTOR (0.39) GSK3BROCK2AURKBPIM1CLK1
SCHEMBL807975 0.81 PRKDC (0.44) PIK3CBPRKDCATRATRIPATM
SCHEMBL807973 0.80 ATM (0.41) PIK3CAPIK3CBPRKDCATRATRIP
SCHEMBL15133606 0.79 MTOR (0.46) ROCK2AURKBCLK4PRKCQROCK1
SCHEMBL1141996 0.78 GSK3B (0.61) GSK3BROCK2AURKBPIM1QPCT
Hydrochloric Acid SCHEMBL1142046 0.76 GSK3B (0.59) GSK3BROCK2AURKBPIM1QPCT
SCHEMBL10070634 0.75 MAPT (0.41) AURKBPIK3CAPIK3CBPRKDCATR
SCHEMBL807826 0.71 PI4KA (0.45) PIK3CAPIK3CB
SCHEMBL15131796 0.71 MTOR (0.49) AURKBCLK4PIK3CAPIK3CBPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012034526-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2012-03-22 WO disclosed