SCHEMBL8080392

SCHEMBL8080392

Cc1cccc(-c2c3c(cc4ccc5c(c24)OCO5)C(=O)NC3=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
NR3C2 P08235 1/20 0.40
CDK2 P24941 4/20 0.39
CHEK1 O14757 1/20 0.39
WEE1 P30291 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
AURKA O14965 1/20 0.38
CDK1 P06493 1/20 0.38
CDK4 P11802 1/20 0.38
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
ALOX5 P09917 4/20 0.35
NQO2 P16083 1/20 0.34
MAOB P27338 1/20 0.34
FYN P06241 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085040 0.88 CDK2 (0.39) ALDH1A1CDK2CHEK1WEE1AURKA
SCHEMBL2959109 0.85 ALOX5 (0.48) CDK2ALOX5MEN1KMT2A
SCHEMBL8080585 0.83 ALOX5 (0.53) ALDH1A1HPGDNR3C2CDK2L3MBTL1
SCHEMBL8072614 0.82 CHEK1 (0.40) CDK2CHEK1WEE1GAAAURKA
SCHEMBL8086819 0.81 CDK2 (0.39) CDK2CHEK1WEE1AURKACDK1
SCHEMBL8082093 0.81 CDK2 (0.39) CDK2AURKACDK1CDK4HSP90AA1
SCHEMBL8084885 0.81 PTGS2 (0.44) NR3C2CDK2CHEK1WEE1AURKA
SCHEMBL2960392 0.81 TOP2A (0.48) ALDH1A1HPGDCDK2L3MBTL1CDK4
SCHEMBL8080517 0.80 APP (0.41) ALDH1A1HPGDCDK2CHEK1WEE1
SCHEMBL8072321 0.79 CDK2 (0.43) ALDH1A1HPGDCDK2AURKACDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6030967-A AND/OR LIKE NEUROTROPHIC FACTOR (FOR EXAMPLE, NERVE GROWTH FACTOR (NGF), BRAIN-DERIVED NEUROTROPHIC FACTOR, NEUROTROPHIN-3, AND GLIAL CELL LINE-DERIVED NEUROTROPHIC FACTOR)-LIKE ACTIVITY; OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-02-29 US disclosed