SCHEMBL8081003

SCHEMBL8081003

COC(=O)C[C@@H](NC(=O)OC(C)(C)C)C1CC2CCC(C1)N2C(=O)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 5/20 0.38
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
REN P00797 2/20 0.35
ITGB3 P05106 2/20 0.35
ITGA2B P08514 2/20 0.35
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
BTK Q06187 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
PREP P48147 1/20 0.33
EPHX1 P07099 1/20 0.33
AAK1 Q2M2I8 1/20 0.32
KMT2A Q03164 1/20 0.32
HPGD P15428 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13078578 0.86 CACNA1B (0.37) CACNA1BCTSSCTSKRENITGB3
SCHEMBL10060683 0.83 CYP2D6 (0.38) CACNA1BCTSSCTSKRENCHRM2
SCHEMBL7849129 0.83 CYP2D6 (0.38) CACNA1BCTSSCTSKRENCHRM2
SCHEMBL3806247 0.81 BTK (0.39) CACNA1BCTSSCTSKITGB3ITGA2B
SCHEMBL3751248 0.80 BTK (0.40) CTSSCTSKITGB3ITGA2BCHRM2
SCHEMBL13078813 0.80 CTSK (0.34) CACNA1BCTSSCTSKCHRM2CHRM1
SCHEMBL13078576 0.77 DPP4 (0.37) CACNA1BRENCHRM2CHRM1CHRM3
SCHEMBL13078880 0.77 ELANE (0.34) CACNA1BCTSSCTSKBTKKMT2A
SCHEMBL13078577 0.76 CACNA1B (0.34) CACNA1BRENKMT2ACYP2D6
SCHEMBL13078575 0.75 CTSL (0.46) CACNA1BRENKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037719-A1 NOVEL COMPOUNDS AS DIPEPTIDYL PEPTIDASE IV (DPP IV) INHIBITORS LUPIN LIMITED (IN) 2009-03-26 WO disclosed