SCHEMBL8081895

SCHEMBL8081895

Cc1nn(C)c(C(=O)NCc2c(F)c(F)c(CC(C)(C)C)c(F)c2F)c1Cl

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
KMT2A Q03164 2/20 0.55
GALR3 O60755 1/20 0.55
NR2F2 P24468 1/20 0.55
RAB9A P51151 1/20 0.55
KDM4E B2RXH2 2/20 0.52
ALPL P05186 2/20 0.43
ALPI P09923 1/20 0.43
ALPG P10696 1/20 0.43
GAA P10253 3/20 0.43
ALDH1A1 P00352 7/20 0.41
HPGD P15428 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPT P10636 2/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8079080 0.88 LMNA (0.55) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8079104 0.88 LMNA (0.50) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8083894 0.86 LMNA (0.40) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8079112 0.84 LMNA (0.56) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8083964 0.83 LMNA (0.55) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8083952 0.83 LMNA (0.55) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8069722 0.83 LMNA (0.50) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8079241 0.83 LMNA (0.52) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8069686 0.82 LMNA (0.54) LMNASMN1; SMN2KMT2AGALR3NR2F2
SCHEMBL8079219 0.82 LMNA (0.51) LMNASMN1; SMN2KMT2AGALR3NR2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634403-B1 N-polyhalobenzyl-pyrazole carboxamides endowed with acaricidal and insecticidal activity ISAGRO SPA (IT) 2000-09-13 EP disclosed
US-5541214-A N-polyhalobenzyl-pyrazole carboxamides endowed with acaricidal and insecticidal activity ISAGRO S.P.A. (IT) 1996-07-30 US disclosed
EP-0634403-A1 N-polyhalobenzyl-pyrazole carboxamides endowed with acaricidal and insecticidal activity ISAGRO S.p.A. (IT) 1995-01-18 EP disclosed