SCHEMBL8079112

SCHEMBL8079112

CCCc1c(F)c(F)c(CNC(=O)c2c(Cl)c(C)nn2C)c(F)c1F

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 8/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
RAB9A P51151 4/20 0.56
KMT2A Q03164 2/20 0.56
GALR3 O60755 1/20 0.56
NR2F2 P24468 1/20 0.56
KDM4E B2RXH2 2/20 0.53
GAA P10253 3/20 0.49
ALPL P05186 2/20 0.44
ALPI P09923 1/20 0.44
ALPG P10696 1/20 0.44
ALDH1A1 P00352 6/20 0.42
HPGD P15428 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 3/20 0.40
MAPT P10636 3/20 0.40
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083964 0.94 LMNA (0.55) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8069686 0.93 LMNA (0.54) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8079134 0.87 LMNA (0.53) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8069768 0.87 LMNA (0.48) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8079219 0.85 LMNA (0.51) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8081895 0.84 LMNA (0.55) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8079080 0.84 LMNA (0.55) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8083952 0.84 LMNA (0.55) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8069795 0.83 LMNA (0.49) LMNASMN1; SMN2RAB9AKMT2AGALR3
SCHEMBL8069563 0.83 LMNA (0.52) LMNASMN1; SMN2RAB9AKMT2AGALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634403-B1 N-polyhalobenzyl-pyrazole carboxamides endowed with acaricidal and insecticidal activity ISAGRO SPA (IT) 2000-09-13 EP disclosed
US-5541214-A N-polyhalobenzyl-pyrazole carboxamides endowed with acaricidal and insecticidal activity ISAGRO S.P.A. (IT) 1996-07-30 US disclosed
EP-0634403-A1 N-polyhalobenzyl-pyrazole carboxamides endowed with acaricidal and insecticidal activity ISAGRO S.p.A. (IT) 1995-01-18 EP disclosed