SCHEMBL8082501

SCHEMBL8082501

CC(N=C(N)N)c1ccc(N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.47
HTT P42858 2/20 0.42
ALDH1A1 P00352 4/20 0.39
GRIN2D O15399 3/20 0.39
GRIN3B O60391 3/20 0.39
GRIN1 Q05586 3/20 0.39
GRIN2A Q12879 3/20 0.39
GRIN2B Q13224 3/20 0.39
GRIN2C Q14957 3/20 0.39
GRIN3A Q8TCU5 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NOS3 P29474 4/20 0.39
NOS1 P29475 4/20 0.39
MAPT P10636 3/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HIF1A Q16665 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8079624 0.98 NOS2 (0.46) NOS2HTTALDH1A1GRIN2DGRIN3B
SCHEMBL22180009 0.81 NOS2 (0.46) NOS2HTTGRIN2DGRIN3BGRIN1
SCHEMBL6682638 0.81 NOS2 (0.46) NOS2HTTALDH1A1GRIN2DGRIN3B
SCHEMBL7020087 0.80 NOS2 (0.70) NOS2ALDH1A1NOS3KDM4EHIF1A
SCHEMBL6682071 0.77 NOS2 (0.46) NOS2HTTALDH1A1GRIN2DGRIN3B
SCHEMBL20487491 0.76 CA12 (0.48) NOS2HTTALDH1A1SMN1; SMN2NOS1
Hydrochloric Acid SCHEMBL7327781 0.75 CA12 (0.47) NOS2HTTALDH1A1SMN1; SMN2NOS1
SCHEMBL5955 0.70 MAPT (0.53) NOS2HTTALDH1A1SMN1; SMN2NOS3
SCHEMBL56667 0.69 NOS3 (0.50) HTTALDH1A1NOS3NOS1MAPT
SCHEMBL12122146 0.69 NOS3 (0.50) HTTALDH1A1NOS3NOS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882066-B1 PEPTIDE DERIVATIVES ZENECA LTD (GB) 2000-09-06 EP disclosed
US-6087336-A ANTIINFLAMMATORY AGENT TREATING RHEUMATOID ARTHRITIS ZENECA LIMITED (GB) 2000-07-11 US disclosed
EP-0882066-A1 PEPTIDE DERIVATIVES ZENECA LIMITED (GB) 1998-12-09 EP disclosed
WO-1997031023-A1 PEPTIDE DERIVATIVES ZENECA LIMITED (GB) 1997-08-28 WO disclosed