SCHEMBL8082744

SCHEMBL8082744

Cc1cncc(-c2cnc(C3CCCC3)c(OC=O)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.35
CYP2A6 P11509 1/20 0.32
PIK3CB P42338 1/20 0.31
PRKDC P78527 1/20 0.31
ATM Q13315 1/20 0.31
ATR Q13535 1/20 0.31
ATRIP Q8WXE1 1/20 0.31
CYP11B1 P15538 2/20 0.31
CTPS1 P17812 1/20 0.31
CHRNB1 P11230 2/20 0.31
CHRNB2 P17787 2/20 0.31
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
CHRNB3 Q05901 2/20 0.31
CHRNA4 P43681 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
GCK P35557 1/20 0.31
LRRK2 Q5S007 2/20 0.30
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12044408 0.78 CYP2A6 (0.38) CYP11B2CYP2A6PIK3CBPRKDCATM
SCHEMBL2276825 0.75 ATM (0.44) CYP11B2ATM
SCHEMBL12024920 0.74 CYP11B2 (0.41) CYP11B2PDE10A
SCHEMBL2278188 0.72 CYP11B2 (0.40) CYP11B2CYP2A6CTPS1LRRK2PDE10A
SCHEMBL10133638 0.69 CYP11B2 (0.35) CYP11B2CYP2A6PIK3CBPRKDCATM
SCHEMBL438348 0.67 ATM (0.41) CYP11B2ATMATRCYP11B1PDE10A
SCHEMBL7877414 0.67 ACVR2A (0.38) CYP11B2PIK3CBPRKDCATMATR
SCHEMBL23959742 0.65 CYP11B2 (0.40) CYP11B2CYP2A6
SCHEMBL20345770 0.65 CYP17A1 (0.33) CYP11B2
SCHEMBL27680007 0.63 FDPS (0.43) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020642-A1 PYRIDINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-02-12 WO disclosed