SCHEMBL8083480

SCHEMBL8083480

OCCn1cnc2c(-c3ccc4cc[nH]c4c3)nc(N3CCOCC3)nc21

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.48
PIK3R1 P27986 4/20 0.48
HDAC1 Q13547 13/20 0.47
MTOR P42345 3/20 0.46
PIK3CG P48736 1/20 0.42
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
HDAC3 O15379 9/20 0.41
HDAC4 P56524 9/20 0.41
HDAC7 Q8WUI4 9/20 0.41
HDAC2 Q92769 9/20 0.41
HDAC10 Q969S8 9/20 0.41
HDAC11 Q96DB2 9/20 0.41
HDAC8 Q9BY41 9/20 0.41
HDAC6 Q9UBN7 9/20 0.41
HDAC9 Q9UKV0 9/20 0.41
HDAC5 Q9UQL6 9/20 0.41
ATR Q13535 1/20 0.40
ATRIP Q8WXE1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL944808 0.89 PIK3CA (0.49) PIK3CAPIK3R1HDAC1MTORHDAC3
SCHEMBL12910204 0.88 PIK3CA (0.44) PIK3CAPIK3R1HDAC1MTORPIK3CG
SCHEMBL12910202 0.86 ATR (0.48) PIK3CAPIK3R1HDAC1MTORPIK3CG
SCHEMBL1568565 0.85 PIK3CA (0.53) PIK3CAPIK3R1HDAC1MTORHDAC3
SCHEMBL12910182 0.85 PDE10A (0.48) PIK3CAPIK3R1HDAC1MTORPIK3CG
SCHEMBL12910205 0.85 PIK3CA (0.47) PIK3CAPIK3R1HDAC1HDAC3HDAC4
SCHEMBL1569308 0.82 PIK3CA (0.57) PIK3CAPIK3R1HDAC1MTORPIK3CG
SCHEMBL1570938 0.82 PIK3CA (0.59) PIK3CAPIK3R1HDAC1MTORHDAC3
SCHEMBL12910556 0.82 CSNK1E (0.44) PIK3CAHDAC1MTORHDAC3HDAC4
SCHEMBL12910192 0.80 ALDH1A1 (0.49) PIK3CAHDAC1HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045174-A1 2-MORPHOLINYLPURINES AS INHIBITORS OF PI3K S*BIO PTE LTD (SG) 2009-04-09 WO disclosed