SCHEMBL8083749

SCHEMBL8083749

CS(=O)(=O)C1(c2cc(N)nc(-c3ccc(NC(=O)NCCO)nc3)n2)CCCC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.37
MAPK1 P28482 1/20 0.36
PIK3CA P42336 7/20 0.36
MTOR P42345 2/20 0.36
PIK3CD O00329 7/20 0.35
PIK3CB P42338 3/20 0.35
PIK3CG P48736 3/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PIK3R1 P27986 1/20 0.33
F10 P00742 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091865 0.91 MAPK1 (0.42) EPHX2MAPK1PIK3CAMTORPIK3CD
SCHEMBL8090668 0.89 PIK3CA (0.35) MAPK1PIK3CAMTORPIK3CDPIK3CB
SCHEMBL8083676 0.88 PIK3CA (0.46) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL8092989 0.86 PIK3CA (0.46) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL8083702 0.83 PIK3CD (0.41) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL8083631 0.81 PIK3CD (0.41) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL8099345 0.81 PIK3CD (0.44) PIK3CAMTORPIK3CDPIK3CGRAB9A
SCHEMBL3935608 0.80 PIK3CA (0.58) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL8092066 0.80 PIK3CA (0.44) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL8083872 0.80 PIK3CA (0.50) PIK3CAMTORPIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed