SCHEMBL8084236

SCHEMBL8084236

CC(=O)OC1(C)C(Oc2ccc(O)nn2)c2cc(C#N)ccc2OC1(C)C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
ABCC9 O60706 5/20 0.38
CYP3A4 P08684 2/20 0.37
ALOX15 P16050 1/20 0.37
ABCB1 P08183 10/20 0.37
KCNE1 P15382 3/20 0.35
KCNQ1 P51787 3/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
KCND3 Q9UK17 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323808 0.89 KDM4E (0.37) KDM4EABCC9CYP3A4ABCB1KCNE1
SCHEMBL7273801 0.85 ABCC9 (0.39) KDM4EABCC9ABCB1
SCHEMBL8090760 0.82 KDM4E (0.40) KDM4EABCC9CYP3A4ALOX15ABCB1
SCHEMBL8085191 0.78 KCNE1 (0.38) KDM4EABCC9CYP3A4ABCB1KCNE1
SCHEMBL8076898 0.78 KCNE1 (0.38) KDM4EABCC9CYP3A4ABCB1KCNE1
SCHEMBL8090688 0.77 KCNE1 (0.38) KDM4EABCC9CYP3A4ABCB1KCNE1
SCHEMBL8085269 0.77 ABCC9 (0.36) KDM4EABCC9CYP3A4ABCB1KCNE1
SCHEMBL8085394 0.77 ABCC9 (0.36) KDM4EABCC9CYP3A4ABCB1KCNE1
SCHEMBL9443454 0.77 KDM4E (0.41) KDM4EABCC9CYP3A4ALOX15ABCB1
SCHEMBL7331226 0.77 ABCC9 (0.46) KDM4EABCC9CYP3A4ALOX15ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed