SCHEMBL8084243

SCHEMBL8084243

CC1(C)Oc2ccc([N+](=O)[O-])cc2C(n2cc(N)ccc2=O)C1(C)O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.33
AKR1B1 P15121 2/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
ALDH1A1 P00352 4/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HIF1A Q16665 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CYP3A4 P08684 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 3/20 0.31
GAA P10253 1/20 0.31
THRB P10828 1/20 0.31
TSHR P16473 1/20 0.31
LMNA P02545 2/20 0.30
RAB9A P51151 1/20 0.30
TLR9 Q9NR96 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8077027 0.91 ALDH1A1 (0.36) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8174422 0.88 HIF1A (0.34) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8076915 0.88 ALDH1A1 (0.34) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8088875 0.86 ABCC9 (0.34) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8090050 0.86 MEN1 (0.39) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8090465 0.85 MAPT (0.34) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8088428 0.84 SMN1; SMN2 (0.40) MEN1KMT2AALDH1A1CYP3A4TDP1
SCHEMBL8084249 0.83 HIF1A (0.35) ABCC9AKR1B1MEN1KMT2AALDH1A1
SCHEMBL8084634 0.81 ABCC9 (0.40) ABCC9LMNA
SCHEMBL8088701 0.81 ABCC9 (0.47) ABCC9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed