SCHEMBL8084403

SCHEMBL8084403

COCC(=C(C(=O)O)c1ccccc1)c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.54
ESR2 Q92731 3/20 0.49
AKR1C2 P52895 1/20 0.46
AKR1C1 Q04828 1/20 0.46
AKR1C3 P42330 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084402 1.00 PTGS2 (0.54) PTGS2ESR2AKR1C2AKR1C1AKR1C3
SCHEMBL5072268 0.86 PTGS2 (0.53) PTGS2ESR2
SCHEMBL3988166 0.86 PTGS2 (0.53) PTGS2ESR2
SCHEMBL3988162 0.86 PTGS2 (0.53) PTGS2ESR2
SCHEMBL5338840 0.85 ESR2 (0.58) PTGS2ESR2
SCHEMBL5338833 0.85 ESR2 (0.58) PTGS2ESR2
SCHEMBL5340116 0.79 ESR2 (0.45) PTGS2ESR2
SCHEMBL5340111 0.79 ESR2 (0.45) PTGS2ESR2
SCHEMBL8425841 0.78 PTGS2 (0.50) PTGS2ESR2
SCHEMBL5343680 0.78 ESR2 (0.44) PTGS2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882015-B1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2000-12-27 EP claimed
US-5733909-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT MERCK FROSST CANADA, INC. (CA) 1998-03-31 US claimed
EP-0882015-B1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2000-12-27 EP disclosed
US-5733909-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT MERCK FROSST CANADA, INC. (CA) 1998-03-31 US disclosed