SCHEMBL8085859

SCHEMBL8085859

CC(=O)NC1CCNC(c2ccccc2)C1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
FASN P49327 1/20 0.43
ATM Q13315 2/20 0.42
ALOX15 P16050 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM1A O60341 5/20 0.40
HPGD P15428 1/20 0.38
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
CISD1 Q9NZ45 1/20 0.37
SLC6A2 P23975 1/20 0.37
MAOB P27338 1/20 0.37
HTR1B P28222 1/20 0.37
HTR2A P28223 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16401194 0.88 KDM1A (0.40) SMN1; SMN2NPSR1KDM1AHPGDCISD1
SCHEMBL22032415 0.88 KDM1A (0.40) SMN1; SMN2NPSR1KDM1AHPGDCISD1
SCHEMBL22032451 0.88 KDM1A (0.40) SMN1; SMN2NPSR1KDM1AHPGDCISD1
SCHEMBL25619917 0.82 ALDH1A1 (0.43) SMN1; SMN2ATMALDH1A1HPGDKDM4E
SCHEMBL25053373 0.81 KDM1A (0.57) KDM1AMAOB
SCHEMBL22086333 0.81 KDM1A (0.57) KDM1AMAOB
SCHEMBL29116029 0.81 KDM1A (0.57) KDM1AMAOB
SCHEMBL29373513 0.81 KDM1A (0.57) KDM1AMAOB
SCHEMBL30141966 0.80 KDM1A (0.45) KDM1ACISD1SLC6A2MAOBHTR1B
SCHEMBL16403103 0.80 KDM1A (0.45) KDM1ACISD1SLC6A2MAOBHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080743-A AS CHEMICAL INTERMEIDATES FOR PREPARING DRUGS NOVARTIS AG (CH) 2000-06-27 US disclosed
EP-0853617-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES Novartis AG (CH) 1998-07-22 EP disclosed
WO-1997008155-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES NOVARTIS AG (CH) 1997-03-06 WO disclosed