SCHEMBL8085883

SCHEMBL8085883

CCCCCOc1cccc2c1CN(CCc1ccc(O)cc1)C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.47
S1PR5 Q9H228 2/20 0.45
HRH3 Q9Y5N1 2/20 0.44
PTGER4 P35408 1/20 0.42
PTGER2 P43116 1/20 0.42
NR5A1 Q13285 1/20 0.42
ESR1 P03372 2/20 0.40
ADRA2A P08913 2/20 0.40
ADORA3 P0DMS8 2/20 0.40
TACR2 P21452 2/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TP53 P04637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
SHBG P04278 1/20 0.40
CYP3A4 P08684 1/20 0.40
HSPD1 P10809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085031 0.77 CNR2 (0.56) CNR2ALDH1A1LMNA
SCHEMBL8089406 0.77 CNR2 (0.70) CNR2S1PR5ESR1ADRA2AADORA3
SCHEMBL8078040 0.70 CNR2 (0.69) CNR2ESR1ADRA2AADORA3TACR2
SCHEMBL8185348 0.69 S1PR5 (0.60) S1PR5HRH3ADRA2ATP53ADRA2B
SCHEMBL8191897 0.69 HRH3 (0.66) S1PR5HRH3ADRA2AKDM4EADRA2B
SCHEMBL8184976 0.69 S1PR5 (0.60) S1PR5HRH3ADRA2ATP53ADRA2B
SCHEMBL8086144 0.68 ESR1 (0.40) CNR2NR5A1ESR1ADRA2AADORA3
SCHEMBL22692751 0.68 S1PR5 (0.54) S1PR5HRH3SLC6A4
SCHEMBL29174136 0.67 NR5A1 (0.77) NR5A1ESR1ADRA2AADORA3TACR2
SCHEMBL8187259 0.66 HRH3 (0.58) S1PR5HRH3ADRA2AKDM4EADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017919-A Compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2000-01-25 US disclosed
EP-0887340-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco Inc. (JP) 1998-12-30 EP disclosed