SCHEMBL8185348

SCHEMBL8185348

CCCCCCCCCCCCCCOc1cccc2c1CCN(C)C2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 2/20 0.60
HRH3 Q9Y5N1 3/20 0.56
ADRA2A P08913 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
HTR1A P08908 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
BRD9 Q9H8M2 1/20 0.45
PRMT5 O14744 1/20 0.44
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
ACACB O00763 1/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
ABHD6 Q9BV23 1/20 0.42
DRD2 P14416 1/20 0.42
DRD1 P21728 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8190334 0.94 HRH3 (0.58) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8190341 0.90 HRH3 (0.56) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8184976 0.89 S1PR5 (0.60) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8190422 0.85 HRH3 (0.52) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL10571355 0.85 HRH3 (0.54) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8189400 0.85 HRH3 (0.49) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8187058 0.84 ADRA2A (0.57) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8187259 0.83 HRH3 (0.58) S1PR5HRH3ADRA2AADRA2BADRA2C
SCHEMBL8176552 0.83 S1PR5 (0.60) S1PR5HRH3ADRA2AADRA2BADRA2C
Ammonia Solution, Strong SCHEMBL8185454 0.83 ADRA2A (0.56) S1PR5HRH3ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096752-A Method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives HEINONEN PETRI (FI) 2000-08-01 US disclosed
US-5912342-A SYNTHESIS OF COMBINATORIAL LIBRARIES BY COMPUTER CONTROLLED ROBOT HEINONEN PETRI (FI) 1999-06-15 US disclosed
EP-0910562-A2 A METHOD FOR THE PREPARATION OF TERTIARY AMINES, A COMPOUND USEFUL THEREFOR AND ALPHA-2-RECEPTOR ACTIVE TETRAHYDROISOQUINOLINE DERIVATIVES Oy Juvantia Pharma Ltd (FI) 1999-04-28 EP disclosed
WO-1998051672-A2 A METHOD FOR THE PREPARATION OF TERTIARY AMINES, A COMPOUND USEFUL THEREFOR AND ALPHA-2-RECEPTOR ACTIVE TETRAHYDROISOQUINOLINE DERIVATIVES OY JUVANTIA PHARMA LTD. (FI) 1998-11-19 WO disclosed