SCHEMBL8086903

SCHEMBL8086903

COc1nc2cc(Br)cc(CNC(=O)C(=O)O)c2nc1OC

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 2/20 0.35
TP53 P04637 2/20 0.35
MAPT P10636 4/20 0.35
TTR P02766 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
TSHR P16473 2/20 0.33
NQO2 P16083 2/20 0.33
HSD17B10 Q99714 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8078878 0.86 GPR35 (0.41) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
Acetoacetic Acid SCHEMBL27440708 0.84 KDM4E (0.32) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL27463844 0.82 KDM4E (0.38) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL8085969 0.77 NQO2 (0.40) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL8183610 0.77 MEN1 (0.32) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL8086079 0.75 LATS1 (0.35) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL5973164 0.75 NQO2 (0.41) ALDH1A1MAPTNQO2
SCHEMBL27444188 0.75 SLC7A5 (0.40) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL8498410 0.74 NQO2 (0.32) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL5973831 0.74 NQO2 (0.40) ALDH1A1MAPTNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080743-A AS CHEMICAL INTERMEIDATES FOR PREPARING DRUGS NOVARTIS AG (CH) 2000-06-27 US disclosed
EP-0853617-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES Novartis AG (CH) 1998-07-22 EP disclosed
WO-1997008155-A1 NOVEL 2,3-DIOXO-1,2,3,4-TETRAHYDRO-QUINOYXALINYL DERIVATIVES NOVARTIS AG (CH) 1997-03-06 WO disclosed