SCHEMBL8087290

SCHEMBL8087290

COc1ccc2c(C)cc(Cl)nc2c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.47
MAPT P10636 4/20 0.45
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NQO2 P16083 6/20 0.41
CYP19A1 P11511 2/20 0.40
NPC1 O15118 2/20 0.39
POLB P06746 1/20 0.39
G6PD P11413 1/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
PDPK1 O15530 1/20 0.39
S1PR1 P21453 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13090541 0.88 LMNA (0.46) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL314537 0.86 ALDH1A1 (0.42) MAPTKDM4EALDH1A1HPGDTSHR
SCHEMBL10099092 0.84 MAPT (0.59) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL5440649 0.83 LMNA (0.59) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL10099061 0.79 KDM4E (0.41) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL4816462 0.78 LMNA (0.53) LMNAMAPTKDM4EALDH1A1TSHR
SCHEMBL8271690 0.76 MAPT (0.43) MAPTKDM4EALDH1A1HPGDTSHR
SCHEMBL2838267 0.76 ALDH1A1 (0.39) MAPTKDM4EALDH1A1HPGDTSHR
SCHEMBL13905092 0.75 LMNA (0.50) LMNAMAPTKDM4EALDH1A1TSHR
SCHEMBL313189 0.74 CSF1R (0.44) LMNAMAPTKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009014730-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2009-01-29 WO disclosed