SCHEMBL8087309

SCHEMBL8087309

CCCCc1ccccc1Cc1ccc(Cc2ccccc2CCCC)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.50
LIPG Q9Y5X9 1/20 0.46
TLR8 Q9NR97 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
KEAP1 Q14145 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
HSD11B1 P28845 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CYSLTR2 Q9NS75 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093734 0.94 HTR2A (0.55) HTR2ALIPGTLR8LMNAHTT
SCHEMBL6547306 0.94 HTR2A (0.59) HTR2ALIPGTLR8CYP3A4CYP2D6
SCHEMBL8086301 0.94 LIPG (0.53) HTR2ALIPGTLR8CYP3A4SLC6A2
SCHEMBL6546225 0.92 HTR2A (0.44) HTR2ALIPGTLR8CYP3A4CYP2D6
SCHEMBL8099212 0.92 HTR2A (0.44) HTR2ALIPGTLR8CYP3A4CYP2D6
SCHEMBL8095272 0.92 LIPG (0.56) HTR2ALIPGTLR8CYP3A4SLC6A2
SCHEMBL8098698 0.92 LIPG (0.56) HTR2ALIPGTLR8CYP3A4SLC6A2
SCHEMBL8100866 0.92 LIPG (0.56) HTR2ALIPGTLR8CYP3A4SLC6A2
SCHEMBL9720016 0.91 KEAP1 (0.56) HTR2ALIPGCYP3A4CYP2D6CYP2C9
SCHEMBL8771661 0.89 HTR2A (0.50) HTR2ALIPGTLR8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed