SCHEMBL8088913

SCHEMBL8088913

CCCC[C@H]1CC[C@H]2[C@@H]3CCc4cc(NS(=O)(=O)O)ccc4[C@H]3CC[C@]12C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 6/20 0.53
ABCC4 O15439 2/20 0.52
ABCC1 P33527 1/20 0.52
LMNA P02545 5/20 0.50
ESR1 P03372 5/20 0.50
MAPT P10636 3/20 0.50
KMT2A Q03164 3/20 0.50
PGR P06401 2/20 0.50
AR P10275 2/20 0.50
MEN1 O00255 2/20 0.50
CYP3A4 P08684 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
POLB P06746 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CHRM1 P11229 1/20 0.50
TBXA2R P21731 1/20 0.50
PTGS1 P23219 1/20 0.50
ATM Q13315 1/20 0.50
PDE3A Q14432 1/20 0.50
USP2 O75604 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3908652 0.86 ABCC1 (0.70) STSABCC4ABCC1LMNAESR1
SCHEMBL5158101 0.83 ESR1 (0.70) STSLMNAESR1MAPTKMT2A
SCHEMBL17515286 0.82 ABCC4 (0.56) STSABCC4ABCC1LMNAESR1
SCHEMBL7612623 0.81 LMNA (0.70) STSABCC4ABCC1LMNAESR1
SCHEMBL11783196 0.81 STS (0.69) STSLMNAESR1MAPTKMT2A
SCHEMBL11788270 0.80 STS (0.67) STSLMNAESR1MAPTKMT2A
SCHEMBL11780732 0.80 STS (0.67) STSLMNAESR1MAPTKMT2A
SCHEMBL17817385 0.80 STS (0.67) STSLMNAESR1MAPTKMT2A
SCHEMBL17515288 0.79 ABCC1 (0.58) STSABCC4ABCC1LMNAESR1
SCHEMBL7096088 0.79 ESR1 (0.68) STSABCC4ABCC1LMNAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042354-A2 ESTRONE SULFAMATE INHIBITORS OF ESTRONE SULFATASE, AND ASSOCIATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE SRI INTERNATIONAL (US) 2000-10-11 EP disclosed
WO-1999033858-A2 ESTRONE SULFAMATE INHIBITORS OF ESTRONE SULFATASE, AND ASSOCIATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE SRI INTERNATIONAL (US) 1999-07-08 WO disclosed