SCHEMBL8089328

SCHEMBL8089328

NC(C(=O)N(CCc1ccc(Cl)cc1)c1cccc(O)c1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GLI1 P08151 2/20 0.40
GLI2 P10070 2/20 0.40
PTGIR P43119 1/20 0.40
OPRK1 P41145 9/20 0.39
OPRM1 P35372 8/20 0.37
OPRD1 P41143 8/20 0.37
DRD2 P14416 4/20 0.37
DRD3 P35462 4/20 0.37
NLRP3 Q96P20 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KYNU Q16719 1/20 0.36
ALOX5 P09917 1/20 0.35
LMNA P02545 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3646622 0.91 PTGIR (0.41) GLI1GLI2PTGIRMEN1KMT2A
SCHEMBL8082608 0.86 TACR1 (0.43) GLI1GLI2OPRK1NLRP3MEN1
SCHEMBL3645986 0.83 TRPM8 (0.41) GLI1GLI2
SCHEMBL3650041 0.83 PTGIR (0.41) GLI1GLI2PTGIROPRM1OPRD1
SCHEMBL3645320 0.83 CETP (0.42) PTGIROPRK1OPRM1OPRD1DRD2
SCHEMBL3648054 0.82 PTGIR (0.40) GLI1GLI2PTGIROPRM1OPRD1
SCHEMBL3641635 0.81 TACR1 (0.42) MEN1KMT2A
SCHEMBL3645573 0.79 PTGIR (0.43) PTGIRMEN1KMT2A
SCHEMBL3645744 0.78 OPRK1 (0.43) OPRK1OPRM1OPRD1DRD2DRD3
SCHEMBL3645748 0.78 OPRK1 (0.43) OPRK1OPRM1OPRD1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016087-A1 MONOAMIDE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed