SCHEMBL8089481

SCHEMBL8089481

C[C@H]1Cc2cc(OC3CCCCO3)ccc2[C@H]2CC[C@]3(C)C(=C(F)F)CC[C@H]3[C@@H]21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.52
HRH3 Q9Y5N1 6/20 0.45
STS P08842 2/20 0.36
MAPT P10636 4/20 0.35
LMNA P02545 2/20 0.35
ESR1 P03372 2/20 0.35
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
GAA P10253 1/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP2C9 P11712 2/20 0.33
ABCC4 O15439 1/20 0.33
ABCC1 P33527 1/20 0.33
SLCO1B1 Q9Y6L6 1/20 0.33
HSD17B1 P14061 1/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8081744 0.87 HSD11B1 (0.52) HSD11B1HRH3STSMAPTLMNA
SCHEMBL13216951 0.87 HSD11B1 (0.52) HSD11B1HRH3STSMAPTLMNA
SCHEMBL12968193 0.86 HSD11B1 (0.50) HSD11B1HRH3STSMAPTLMNA
SCHEMBL1659341 0.86 HSD11B1 (0.50) HSD11B1HRH3STSMAPTLMNA
SCHEMBL5270661 0.85 HSD11B1 (0.51) HSD11B1HRH3STSMAPTLMNA
SCHEMBL7827752 0.85 HSD11B1 (0.69) HSD11B1STSMAPTLMNAESR1
SCHEMBL7830895 0.85 HSD11B1 (0.69) HSD11B1STSMAPTLMNAESR1
SCHEMBL1657796 0.83 HSD11B1 (0.49) HSD11B1HRH3STSMAPTLMNA
SCHEMBL5274231 0.82 HSD11B1 (0.46) HSD11B1HRH3STSMAPTLMNA
SCHEMBL5273029 0.80 HSD11B1 (0.55) HSD11B1HRH3STSMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136800-A STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 2000-10-24 US disclosed
US-6018062-A SUCH AS 17-DIFLUOROMETHYLENE-ESTRA-1,3,5(10)-TRIEN-3-OL; USE AS ANTIOXIDANTS AND VASCULOPROTECTIVE AGENTS AS THEY CAUSE VASODILATOR NITROGEN OXIDE RELEASE AND PREVENT OXIDATION OF LDL CHOLESTEROL SCHERING AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed