SCHEMBL8081744

SCHEMBL8081744

C[C@H]1Cc2cc(OC3CCCCO3)ccc2[C@H]2CC[C@]3(C)C(=O)CC[C@H]3[C@@H]21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.52
MAPT P10636 3/20 0.47
LMNA P02545 2/20 0.47
HSD17B1 P14061 2/20 0.47
RECQL P46063 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 2/20 0.46
STS P08842 8/20 0.45
ESR1 P03372 2/20 0.44
ESR2 Q92731 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
ABCC4 O15439 1/20 0.44
CYP2C9 P11712 1/20 0.44
ABCC1 P33527 1/20 0.44
SLCO1B1 Q9Y6L6 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13216951 1.00 HSD11B1 (0.52) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL11688245 0.89 HSD11B1 (0.51) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL5270661 0.88 HSD11B1 (0.51) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL8089481 0.87 HSD11B1 (0.52) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL1657796 0.86 HSD11B1 (0.49) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL1659341 0.85 HSD11B1 (0.50) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL12968193 0.85 HSD11B1 (0.50) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL1657830 0.84 HSD11B1 (0.69) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL7830892 0.84 HSD11B1 (0.69) HSD11B1MAPTLMNAHSD17B1RECQL
SCHEMBL14421698 0.82 HSD17B1 (0.67) MAPTLMNAHSD17B1RECQLSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136800-A STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 2000-10-24 US disclosed
US-6018062-A SUCH AS 17-DIFLUOROMETHYLENE-ESTRA-1,3,5(10)-TRIEN-3-OL; USE AS ANTIOXIDANTS AND VASCULOPROTECTIVE AGENTS AS THEY CAUSE VASODILATOR NITROGEN OXIDE RELEASE AND PREVENT OXIDATION OF LDL CHOLESTEROL SCHERING AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed