SCHEMBL8089533

SCHEMBL8089533

CC1(C)CCSc2c(C=O)cccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 7/20 0.34
RARB P10826 7/20 0.34
RARG P13631 7/20 0.34
ERN1 O75460 2/20 0.33
TLR2 O60603 1/20 0.33
TLR1 Q15399 1/20 0.33
TLR6 Q9Y2C9 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RXRA P19793 2/20 0.33
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
CYP2A6 P11509 1/20 0.31
CA1 P00915 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6350746 0.75 MEN1 (0.34) RARARARBRARGERN1TLR2
SCHEMBL6032597 0.75 RARA (0.32) RARARARBRARGPTGS1PTGS2
SCHEMBL9092316 0.74 TP53 (0.41) RARARARBRARGERN1TLR2
SCHEMBL7134583 0.72 PTGS1 (0.46) RARARARBRARGPTGS1PTGS2
SCHEMBL6032638 0.72 RARA (0.30) RARARARBRARGPTGS1PTGS2
SCHEMBL27807579 0.71 MEN1 (0.37) ERN1TLR2TLR1TLR6MEN1
SCHEMBL8647409 0.70 ALDH1A1 (0.31) ALDH1A1
SCHEMBL6339231 0.70 RARA (0.33) RARARARBRARG
SCHEMBL6344037 0.69 MEN1 (0.34) RARARARBRARGERN1TLR2
SCHEMBL17918163 0.69 CES1 (0.40) MEN1LMNATHRBBLMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740665-B1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN SALES INC (US) 2000-12-06 EP disclosed
EP-0740665-A1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES Allergan (US) 1996-11-06 EP disclosed
US-5519150-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN (US) 1996-05-21 US disclosed
WO-1995019973-A2 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN (US) 1995-07-27 WO disclosed
US-5420295-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN, INC. (US) 1995-05-30 US disclosed