SCHEMBL8089568

SCHEMBL8089568

CCC1(CC)CCOc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.41
ICAM1 P05362 1/20 0.41
ITGAL P20701 1/20 0.41
MAP3K14 Q99558 1/20 0.40
NR3C1 P04150 1/20 0.39
LMNA P02545 2/20 0.38
CRHBP P24387 2/20 0.38
CRHR2 Q13324 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 2/20 0.36
KIF11 P52732 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6124712 0.90 MAP3K14 (0.39) ITGB2ICAM1ITGALMAP3K14NR3C1
SCHEMBL5173976 0.87 NR3C1 (0.38) ITGB2ICAM1ITGALMAP3K14NR3C1
SCHEMBL5174599 0.86 NR3C1 (0.38) ITGB2ICAM1ITGALMAP3K14NR3C1
SCHEMBL25871757 0.81 ITGB2 (0.41) ITGB2ICAM1ITGALMAP3K14LMNA
SCHEMBL5467643 0.80 NR3C1 (0.41) MAP3K14NR3C1SMN1; SMN2KMT2AKIF11
SCHEMBL5173909 0.79 KMT2A (0.34) ITGB2ICAM1ITGALMAP3K14NR3C1
SCHEMBL17295888 0.79 MAP3K14 (0.63) ITGB2ICAM1ITGALMAP3K14LMNA
SCHEMBL19130581 0.79 MAP3K14 (0.63) ITGB2ICAM1ITGALMAP3K14LMNA
SCHEMBL7671149 0.77 ITGB2 (0.38) ITGB2ICAM1ITGALMAP3K14LMNA
SCHEMBL8089535 0.77 MAP3K14 (0.47) MAP3K14NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740665-B1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN SALES INC (US) 2000-12-06 EP disclosed
EP-0740665-A1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES Allergan (US) 1996-11-06 EP disclosed
US-5519150-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN (US) 1996-05-21 US disclosed
WO-1995019973-A2 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN (US) 1995-07-27 WO disclosed
US-5420295-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN, INC. (US) 1995-05-30 US disclosed