SCHEMBL8089691

SCHEMBL8089691

CNC1CC=CC2CN(c3c(F)cc4c(=O)c(C(=O)O)cn(C5CC5)c4c3F)CC21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 6/20 0.49
TOP2B Q02880 6/20 0.49
ALDH1A1 P00352 4/20 0.49
POLB P06746 2/20 0.49
OPRM1 P35372 2/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
OPRD1 P41143 1/20 0.49
KCNH2 Q12809 6/20 0.48
KDM4E B2RXH2 3/20 0.47
HPGD P15428 3/20 0.47
HSD17B10 Q99714 2/20 0.47
PRKD3 O94806 1/20 0.47
ALOX15 P16050 1/20 0.47
CLK2 P49760 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083224 0.93 ALDH1A1 (0.59) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL8091231 0.90 KDM4E (0.40) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL9044987 0.89 KDM4E (0.39) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL9095828 0.88 KCNH2 (0.48) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL8089789 0.88 ALDH1A1 (0.54) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL8091252 0.86 KCNH2 (0.49) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL8091158 0.86 KCNH2 (0.54) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL9136070 0.85 ALDH1A1 (0.51) TOP2ATOP2BALDH1A1POLBOPRM1
SCHEMBL8090947 0.85 KDM4E (0.57) TOP2ATOP2BALDH1A1KDM4EHPGD
SCHEMBL9779832 0.84 ALDH1A1 (0.53) TOP2ATOP2BALDH1A1POLBOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed
US-5556979-A ANIMAL FEEDS BAYER AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed