SCHEMBL8091231

SCHEMBL8091231

CNC1CC=CC2CN(c3c(F)cc4c(=O)c(C(=O)O)cn(C5CC5F)c4c3F)CC21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.40
ALDH1A1 P00352 7/20 0.40
HPGD P15428 6/20 0.40
HSD17B10 Q99714 5/20 0.40
POLB P06746 3/20 0.40
OPRM1 P35372 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
OPRD1 P41143 1/20 0.40
PMP22 Q01453 1/20 0.40
LMNA P02545 2/20 0.39
ALB P02768 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
KCNH2 Q12809 3/20 0.38
TOP2A P11388 3/20 0.38
TOP2B Q02880 3/20 0.38
AADAT Q8N5Z0 2/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083017 0.93 ALDH1A1 (0.49) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL8089691 0.90 TOP2A (0.49) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL9047385 0.90 KDM4E (0.32) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL8091409 0.89 KDM4E (0.40) KDM4EALDH1A1HPGDHSD17B10POLB
Hydrochloric Acid SCHEMBL8089805 0.85 KCNH2 (0.43) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL8083224 0.83 ALDH1A1 (0.59) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL9047303 0.83 ALDH1A1 (0.39) KDM4EALDH1A1HPGDPOLBOPRM1
SCHEMBL9044987 0.80 KDM4E (0.39) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL9043731 0.80 KDM4E (0.33) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9053681 0.80 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed