SCHEMBL8090489

SCHEMBL8090489

CC(=O)Nc1cc(Br)cn(C2c3cc(C#N)ccc3OC(C)(C)C2(C)O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ABCC9 O60706 8/20 0.38
ABCB1 P08183 4/20 0.37
ABCC8 Q09428 2/20 0.36
KCNJ11 Q14654 2/20 0.36
KCNJ8 Q15842 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 1/20 0.36
LMNA P02545 1/20 0.36
KCNE1 P15382 3/20 0.36
KCNQ1 P51787 3/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
KMT2A Q03164 1/20 0.36
KCND3 Q9UK17 1/20 0.36
DRD2 P14416 3/20 0.35
DRD3 P35462 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085232 0.90 ABCC9 (0.42) KDM4EABCC9DRD2DRD3
SCHEMBL8085004 0.87 ABCC9 (0.41) KDM4EABCC9ABCB1ABCC8KCNJ11
SCHEMBL8085192 0.86 DRD2 (0.40) KDM4EABCC9ABCB1ABCC8KCNJ11
SCHEMBL8088939 0.85 ABCC9 (0.40) KDM4EABCC9ABCB1ABCC8KCNJ11
SCHEMBL8076903 0.85 ABCC9 (0.39) KDM4EABCC9ABCB1ABCC8KCNJ11
SCHEMBL8090757 0.85 GAA (0.34) ABCC9CYP1A2MEN1KMT2A
SCHEMBL8085315 0.83 DRD2 (0.44) KDM4EABCC9ABCB1DRD2DRD3
SCHEMBL8090533 0.83 ABCC9 (0.52) KDM4EABCC9ABCB1ABCC8KCNJ11
SCHEMBL8085345 0.82 DRD2 (0.42) KDM4EABCC9ABCB1ABCC8KCNJ11
SCHEMBL8088505 0.82 ABCC9 (0.42) KDM4EABCC9ABCB1ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed