SCHEMBL8090574

SCHEMBL8090574

CS(=O)(=O)Cc1cc(N)nc(-c2ccc(NC(=O)c3ccno3)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTOR P42345 5/20 0.51
PIK3CA P42336 6/20 0.47
PIK3CD O00329 6/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.43
MAPK14 Q16539 1/20 0.42
PYGM P11217 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ESR1 P03372 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
ESR2 Q92731 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR2A P28223 1/20 0.38
BACE1 P56817 1/20 0.38
KDM4C Q9H3R0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096450 0.89 KMT2A (0.53) MTORPIK3CAPIK3CDKMT2AMEN1
SCHEMBL8111517 0.84 PTPN1 (0.52) KMT2AMEN1ALDH1A1ESR1POLB
SCHEMBL3065746 0.82 MTOR (0.75) MTORPIK3CAPIK3CDPOLB
SCHEMBL11925797 0.81 PIK3CA (0.49) MTORPIK3CAPIK3CDKMT2AMEN1
SCHEMBL8109642 0.81 PIK3CA (0.49) MTORPIK3CAPIK3CDKMT2AMEN1
SCHEMBL3055635 0.80 PIK3CA (0.73) MTORPIK3CAPIK3CD
SCHEMBL8215041 0.80 PIK3CA (0.66) MTORPIK3CAPIK3CDKMT2AMEN1
SCHEMBL8099295 0.80 CYP3A4 (0.53) KMT2AMEN1ALDH1A1POLBMAPT
SCHEMBL8093349 0.79 PIK3CD (0.48) MTORPIK3CAPIK3CDKMT2AMEN1
SCHEMBL8099372 0.79 PIK3CA (0.48) MTORPIK3CAPIK3CDKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007749-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed