SCHEMBL8096450

SCHEMBL8096450

CS(=O)(=O)Cc1cc(N)nc(-c2cccc(NC(=O)c3ccno3)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MTOR P42345 3/20 0.49
HTT P42858 1/20 0.44
MAPT P10636 1/20 0.44
MEN1 O00255 2/20 0.43
RXFP2 Q8WXD0 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PIK3CA P42336 4/20 0.40
PIK3CD O00329 2/20 0.39
MAPK14 Q16539 1/20 0.39
PARP1 P09874 1/20 0.39
CA2 P00918 1/20 0.39
HDAC1 Q13547 1/20 0.39
FGFR3 P22607 1/20 0.38
KDR P35968 1/20 0.38
ATR Q13535 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090574 0.89 MTOR (0.51) KMT2AMTORMAPTMEN1PIK3CA
SCHEMBL8102170 0.82 CA2 (0.49) KMT2AMAPTMEN1PIK3CAPIK3CD
SCHEMBL3059619 0.81 PIK3CA (0.67) MTORPIK3CAPIK3CDATR
SCHEMBL8111517 0.75 PTPN1 (0.52) KMT2AMAPTMEN1
SCHEMBL3065746 0.73 MTOR (0.75) MTORPIK3CAPIK3CDATR
SCHEMBL8213853 0.73 POLB (0.48) KMT2AMTORMAPTMEN1PIK3CA
SCHEMBL6643138 0.73 HDAC1 (0.66) KMT2AHTTMAPTMEN1RXFP2
SCHEMBL8205071 0.72 PIK3CA (0.54) KMT2AMTORMAPTMEN1RXFP1
SCHEMBL8099295 0.71 CYP3A4 (0.53) KMT2AMAPTMEN1
SCHEMBL3055635 0.70 PIK3CA (0.73) MTORPIK3CAPIK3CDATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007749-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed