SCHEMBL8099372

SCHEMBL8099372

CS(=O)(=O)Cc1cc(N)nc(-c2ccc(NC(=O)C(N)=O)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.48
PIK3CD O00329 7/20 0.48
MTOR P42345 5/20 0.48
ALDH1A1 P00352 5/20 0.40
MEN1 O00255 4/20 0.40
MAPT P10636 4/20 0.40
HPGD P15428 4/20 0.40
KMT2A Q03164 4/20 0.40
KDM4E B2RXH2 3/20 0.40
RXFP1 Q9HBX9 2/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.39
F10 P00742 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11925797 0.90 PIK3CA (0.49) PIK3CAPIK3CDMTORALDH1A1MEN1
SCHEMBL8101524 0.86 MEN1 (0.54) PIK3CAPIK3CDMTORALDH1A1MEN1
SCHEMBL8093349 0.86 PIK3CD (0.48) PIK3CAPIK3CDMTORALDH1A1MEN1
SCHEMBL8218782 0.85 PIK3CA (0.54) PIK3CAPIK3CDMTORMEN1MAPT
SCHEMBL8106030 0.85 PIK3CA (0.47) PIK3CAPIK3CDMTORALDH1A1KMT2A
SCHEMBL8205071 0.85 PIK3CA (0.54) PIK3CAPIK3CDMTORALDH1A1MEN1
SCHEMBL8109642 0.85 PIK3CA (0.49) PIK3CAPIK3CDMTORALDH1A1MEN1
SCHEMBL8104043 0.84 PIK3CA (0.45) PIK3CAPIK3CDMTORALDH1A1MEN1
SCHEMBL8214218 0.84 PIK3CA (0.66) PIK3CAPIK3CDMTOR
SCHEMBL8216901 0.84 PIK3CA (0.53) PIK3CAPIK3CDMTORMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007749-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed