SCHEMBL8090958

SCHEMBL8090958

COc1ccc(COc2ccc(CC(CN(CCN(CC(=O)O)CC(=O)O)CC(=O)O)N(CC(=O)O)CC(=O)O)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 9/20 0.52
NPC1 O15118 1/20 0.51
POLB P06746 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MAOB P27338 8/20 0.51
PLA2G4B P0C869 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085932 0.93 LDHA (0.49) FFAR1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL8090970 0.91 MAOB (0.57) FFAR1MAOB
SCHEMBL8099655 0.87 LDHA (0.48) FFAR1NPC1POLBRAB9ASMN1; SMN2
Caloxetic Acid Free Base SCHEMBL8412091 0.86 MAOB (0.43) POLBSMN1; SMN2MAOB
Caloxetic Acid Free Base SCHEMBL92689 0.86 MAOB (0.43) POLBSMN1; SMN2MAOB
Caloxetic Acid Free Base SCHEMBL19667948 0.85 MAOB (0.42) POLBSMN1; SMN2MAOB
Caloxetic Acid Free Base SCHEMBL29375456 0.85 MAOB (0.42) POLBSMN1; SMN2MAOB
Caloxetic Acid Free Base SCHEMBL19667947 0.85 MAOB (0.42) POLBSMN1; SMN2MAOB
SCHEMBL8092343 0.85 MAOB (0.41) FFAR1SMN1; SMN2MAOB
SCHEMBL8099090 0.84 SMN1; SMN2 (0.44) FFAR1NPC1POLBRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6039931-A Derivatized DTPA complexes, pharmaceutical agents containing these compounds, their use, and processes for their production SCHERING AKTIENGESELLSCHAFT (DE) 2000-03-21 US claimed
EP-0405704-B1 DTPA-complexes derivatives, pharmaceutical compositions containing them, their use and process for their preparation SCHERING AG (DE) 1994-12-14 EP claimed
US-6039931-A Derivatized DTPA complexes, pharmaceutical agents containing these compounds, their use, and processes for their production SCHERING AKTIENGESELLSCHAFT (DE) 2000-03-21 US disclosed
US-5798092-A METAL COMPLEXES; CONTRAST AGENTS FOR MEDICAL IMAGING SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-25 US disclosed