SCHEMBL8091018

SCHEMBL8091018

COc1cc2c(cc1OC)C(N)=NCC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.67
KDM4E B2RXH2 4/20 0.67
MAPT P10636 3/20 0.67
ALDH1A1 P00352 2/20 0.67
GAA P10253 1/20 0.67
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C19 P33261 1/20 0.60
HSD17B10 Q99714 1/20 0.60
RAD52 P43351 2/20 0.60
PKM P14618 1/20 0.60
LMNA P02545 2/20 0.55
MAPK10 P53779 2/20 0.51
GLA P06280 1/20 0.51
RCE1 Q9Y256 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17144905 0.81 ALDH1A1 (0.71) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL1148346 0.80 MAOA (1.00) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL11743358 0.79 MAOA (0.67) MAOAKDM4EMAPTALDH1A1GAA
Hydrochloric Acid SCHEMBL10660329 0.79 MAOA (0.96) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL11742117 0.78 KDM4E (0.61) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL1820002 0.77 CYP1A2 (0.72) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL29868545 0.77 CYP1A2 (0.72) MAOAKDM4EMAPTALDH1A1GAA
Hydrochloric Acid SCHEMBL11744933 0.77 KDM4E (0.59) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL23747284 0.76 KDM4E (0.63) MAOAKDM4EMAPTALDH1A1GAA
SCHEMBL8099984 0.76 ALDH1A1 (0.56) KDM4EMAPTALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6063789-A Aminoisoquinolines and aminotheinopyridine derivatives and their use as anti-inflammatory agents ASTRA PHARMACEUTICALS, LTD. (GB) 2000-05-16 US disclosed
CN-1221407-A Aminoisoquinolines and aminothienopyridine derivatives and their use as anti-inflammatory agents ASTRA PHARMA PROD (GB) 1999-06-30 CN disclosed
EP-0892784-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Astra Pharmaceuticals Limited (GB) 1999-01-27 EP disclosed
WO-1997038977-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS ASTRA PHARMACEUTICALS LTD. (GB) 1997-10-23 WO disclosed
US-4127720-A ANTIALLERGENS BRISTOL-MYERS COMPANY (US) 1978-11-28 US disclosed