SCHEMBL8091029

SCHEMBL8091029

O=C(O)c1cn(C2CC2F)c2c(F)c(N3CC4C=CCC(CN=Cc5cccc([N+](=O)[O-])c5)C4C3)c(F)cc2c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 2/20 0.39
TOP2A P11388 2/20 0.39
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 4/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
POLB P06746 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
CYP3A4 P08684 1/20 0.33
PMP22 Q01453 1/20 0.33
KCNH2 Q12809 2/20 0.32
GUSB P08236 1/20 0.32
LMNA P02545 2/20 0.32
PIK3CD O00329 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CG P48736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8089805 0.79 KCNH2 (0.43) TOP2AALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8902318 0.77 KCNH2 (0.52) TOP1TOP2AALDH1A1KDM4EHPGD
SCHEMBL8902323 0.77 KCNH2 (0.52) TOP1TOP2AALDH1A1KDM4EHPGD
SCHEMBL8091231 0.75 KDM4E (0.40) TOP2AALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8903272 0.74 ALDH1A1 (0.49) TOP1TOP2AALDH1A1KDM4EHPGD
SCHEMBL8903277 0.74 ALDH1A1 (0.49) TOP1TOP2AALDH1A1KDM4EHPGD
SCHEMBL8573058 0.74 ALDH1A1 (0.49) TOP1TOP2AALDH1A1KDM4EHPGD
SCHEMBL8091409 0.72 KDM4E (0.40) TOP2AALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8091252 0.72 KCNH2 (0.49) TOP2AALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8091158 0.71 KCNH2 (0.54) TOP2AALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed
US-5556979-A ANIMAL FEEDS BAYER AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed